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Clinical Pharmacokinetics

Issue 1/2021

Content (10 Articles)

Open Access Pharmacokinetics Review Article

Population Pharmacokinetics of Clotting Factor Concentrates and Desmopressin in Hemophilia

Tim Preijers, Lisette M. Schütte, Marieke J. H. A. Kruip, Marjon H. Cnossen, Frank W. G. Leebeek, Reinier M. van Hest, Ron A. A. Mathôt

Pharmacodynamics Review Article

Review of the Pharmacokinetics and Pharmacodynamics of Intravenous Busulfan in Paediatric Patients

Rachael Lawson, Christine E. Staatz, Christopher J. Fraser, Stefanie Hennig

Antibiotic Systematic Review

Can Population Pharmacokinetics of Antibiotics be Extrapolated? Implications of External Evaluations

Yu Cheng, Chen-yu Wang, Zi-ran Li, Yan Pan, Mao-bai Liu, Zheng Jiao

Open Access NSCLC Original Research Article

Influence of Cow’s Milk and Esomeprazole on the Absorption of Erlotinib: A Randomized, Crossover Pharmacokinetic Study in Lung Cancer Patients

G. D. Marijn Veerman, Koen G. A. M. Hussaarts, Robert Peric, Esther Oomen-de Hoop, Kersten D. Landa, Cor H. van der Leest, Suzanna D. Broerse, Hugo B. Rutten, Huub N. A. Belderbos, Christi M. J. Steendam, Marthe S. Paats, Stijn L. W. Koolen, Anne-Marie C. Dingemans, Teun van Gelder, Roelof W. F. van Leeuwen, Joachim G. J. V. Aerts, Ron H. J. Mathijssen

Open Access Schizophrenia Original Research Article

Pharmacokinetics of ASP4345 from Single Ascending-Dose and Multiple Ascending-Dose Phase I Studies

Amit Desai, Lauren Benner, Ruishan Wu, Lev Gertsik, Tolga Uz, Gerard J. Marek, Tong Zhu

Open Access Pharmacokinetics Original Research Article

Population Pharmacokinetic and Pharmacogenetic Analysis of Mitotane in Patients with Adrenocortical Carcinoma: Towards Individualized Dosing

Anyue Yin, Madeleine H. T. Ettaieb, Jesse J. Swen, Liselotte van Deun, Thomas M. A. Kerkhofs, Robert J. H. M. van der Straaten, Eleonora P. M. Corssmit, Hans Gelderblom, Michiel N. Kerstens, Richard A. Feelders, Marelise Eekhoff, Henri J. L. M. Timmers, Antonio D’Avolio, Jessica Cusato, Henk-Jan Guchelaar, Harm R. Haak, Dirk Jan A. R. Moes

Human Immunodeficiency Virus Original Research Article

Older Age is Associated with Higher Dolutegravir Exposure in Plasma and Cerebrospinal Fluid of People Living with HIV

Andrea Calcagno, José Moltó, Alberto Borghetti, Cristina Gervasoni, Maurizio Milesi, Marta Valle, Valeria Avataneo, Chiara Alcantarini, Francesc Pla-Junca, Mattia Trunfio, Antonio D’Avolio, Simona Di Giambenedetto, Dario Cattaneo, Giovanni Di Perri, Stefano Bonora

Open Access Fibromyalgia Original Research Article

Pharmacokinetics of Ampreloxetine, a Norepinephrine Reuptake Inhibitor, in Healthy Subjects and Adults with Attention-Deficit/Hyperactive Disorder or Fibromyalgia Pain

Jitendra Kanodia, Arthur Lo, R. Michael Baldwin, Richard A. Graham, David L. Bourdet

Norethisterone Original Research Article

Drug–Drug Interaction Studies of Elagolix with Oral and Transdermal Low-Dose Hormonal Add-Back Therapy

Ahmed Nader, Nael M. Mostafa, Farah Ali, Mohamad Shebley