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European Journal of Drug Metabolism and Pharmacokinetics

Issue 1/2024

Content (10 Articles)

Original Research Article

Distribution, Metabolism, and Excretion of Cenobamate in Adult, Fetal, Neonatal, and Lactating Rats

Jairam Palamanda, Kelli J. Glenn, Susan M. Melnick

Pharmacokinetics Original Research Article

Pharmacokinetics of 4-Hydroxybenzaldehyde in Normal and Cerebral Ischemia–Reperfusion Injury Rats Based on Microdialysis Technique

Chunping Xu, Jin Feng, Hang Sun, Mingli Yan, Qian Yang, Xiaonan Zhou, Jianguang Yang, Fangyan He, Qing Lin

Ticagrelor Original Research Article

Ticagrelor Steady-State Trough Concentration in Chinese Patients Undergoing Percutaneous Coronary Intervention

ShaoJun Zheng, Qiong Jie, NaiDong Chen, XiJing Chen, YuBing Zhu

Original Research Article

Pharmacokinetic Parameters of Recombinant Human Cyclophilin A in Mice

Anastasiia Kalinina, Elena Grigorieva, Anna Smirnova, Dmitry Kazansky, Ludmila Khromykh

Pharmacokinetics Original Research Article

Mass Balance and Metabolic Pathways of Eliapixant, a P2X3 Receptor Antagonist, in Healthy Male Volunteers

Stefanie Reif, Marcus-Hillert Schultze-Mosgau, Anna Engelen, Isabel Piel, Karsten Denner, Ad Roffel, Renger Tiessen, Stefan Klein, Klaus Francke, Antje Rottmann

Open Access Tramadol Original Research Article

Development, Physicochemical Characteristics and Pharmacokinetics of a New Sustained-Release Bilayer Tablet Formulation of Tramadol with an Immediate-Release Component for Twice-Daily Administration

Naoki Ishitsubo, Shinji Oguro, Hirotoshi Shimahashi, Masato Kawanishi, Takeshi Adachi, Kenji Mitsuda, Nobuyuki Ishibashi

Open Access Hydroxychloroquine Original Research Article

Evaluation of Hydroxychloroquine as a Perpetrator on Cytochrome P450 (CYP) 3A and CYP2D6 Activity with Microdosed Probe Drugs in Healthy Volunteers

Felicitas Stoll, Antje Blank, Gerd Mikus, David Czock, Johanna Weiss, Marleen J. Meyer-Tönnies, Katja S. Gümüs, Mladen Tzvetkov, Jürgen Burhenne, Walter E. Haefeli

Fatty Liver Original Research Article

Comparative Pharmacokinetic Study of Rhubarb Anthraquinones in Normal and Nonalcoholic Fatty Liver Disease Rats

Fang Zhang, Rui Wu, Yanfang Liu, Shu Dai, Xinyan Xue, Xiaohong Gong, Yunxia Li