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European Journal of Drug Metabolism and Pharmacokinetics

Issue 6/2016

Content (20 Articles)

Acknowledgement to Referees

Acknowledgements

Current opinion

Proposing the Use of Partial AUC as an Adjunctive Measure in Establishing Bioequivalence Between Deltoid and Gluteal Administration of Long-Acting Injectable Antipsychotics

Lik Hang N. Lee, Charles Choi, Pavel Gershkovich, Alasdair M. Barr, William G. Honer, Ric M. Procyshyn

Systematic Review

Interaction of Citrus Juices with Cyclosporine: Systematic Review and Meta-Analysis

Kannan Sridharan, Gowri Sivaramakrishnan

Original Research Article

Single Dose Oral and Intravenous Pharmacokinetics and Tissue Distribution of a Novel Hesperetin Derivative MTBH in Rats

Chenlin Shen, Zhengyue Qian, Ruonan Chen, Xiaoming Meng, Tingting Hu, Zhaolin Chen, Yangyang Li, Cheng Huang, Chaojie Hu, Jun Li

Original Research Article

A Physiologically Based Pharmacokinetic Model of Amiodarone and its Metabolite Desethylamiodarone in Rats: Pooled Analysis of Published Data

Jing-Tao Lu, Ying Cai, Feng Chen, Wei-Wei Jia, Zhe-Yi Hu, Yuan-Sheng Zhao

Original Research Article

Investigation of the Interaction Between Human Serum Albumin and Two Drugs as Binary and Ternary Systems

Nooshin Abdollahpour, Vahid Soheili, Mohammad Reza Saberi, Jamshidkhan Chamani

Original Research Article

Pharmacokinetics of Glycopyrronium Following Repeated Once-Daily Inhalation in Healthy Chinese Subjects

Romain Sechaud, Surendra Machineni, Hanns-Christian Tillmann, Hisanori Hara, Xuemei Tan, Rong Zhao, Shuang Ren, Jie Hou

Original Research Article

Effect of Multi Drug Resistance Protein 4 (MRP4) Inhibition on the Pharmacokinetics and Pharmacodynamics of Ciprofloxacin in Normal and Rats with LPS-Induced Inflammation

V. Gangadhara N. V. Prasad, Satyanarayana Achanta, Yathiraja Rao Tammineni, Gopala Reddy Alla, Madhava Rao Thirtham, G. S. Rao

Original Research Article

Effect of 22 Novel Cytochrome P450 2D6 (CYP2D6) Variants Found in the Chinese Population on Hemangeol Metabolism In Vitro

Bingqing Liang, Yunyun Zhan, Xiangxin Huang, Ermin Gu, Dapeng Dai, Jianping Cai, Guoxin Hu

Original Research Article

Prediction of Antimalarial Drug Clearance in Children: A Comparison of Three Different Interspecies Scaling Methods

Iftekhar Mahmood, Anna Cheng, Edward Brauer, Rita Humeniuk

Original Research Article

Pharmacokinetics of Curcumin Diethyl Disuccinate, a Prodrug of Curcumin, in Wistar Rats

Kunan Bangphumi, Chuleeporn Kittiviriyakul, Pasarapa Towiwat, Pornchai Rojsitthisak, Phisit Khemawoot

Original Research Article

Stereoselective Pharmacokinetics of Ketoprofen After Oral Administration of Modified-Release Formulations in Caucasian Healthy Subjects

Marianela Lorier, Laura Magallanes, Manuel Ibarra, Natalia Guevara, Marta Vázquez, Pietro Fagiolino

Original Research Article

Intestinal Permeability of β-Lapachone and Its Cyclodextrin Complexes and Physical Mixtures

Victor Mangas-Sanjuan, Jorge Gutiérrez-Nieto, Magdalena Echezarreta-López, Isabel González-Álvarez, Marta González-Álvarez, Vicente-Germán Casabó, Marival Bermejo, Mariana Landin

Original Research Article

Enhancement of Dissolution Rate and Intestinal Stability of Clopidogrel Hydrogen Sulfate

Dina E. Bali, Mohamed A. Osman, Gamal M. El Maghraby

Original Research Article

Presence of an H+/Quinidine Antiport System in Madin–Darby Canine Kidney Cells

Miki Fukao, Eri Kondo, Hiroki Nishino, Ryutaro Hattori, Asuka Horie, Yukiya Hashimoto

Original Research Article

Effect of Ginkgo Leaf Tablets on the Pharmacokinetics of Amlodipine in Rats

Rong Wang, Hai Zhang, Sen Sun, Yuanyuan Wang, Yifeng Chai, Yongfang Yuan

Short Communication

Angiotensin Receptor Blocker Losartan Inhibits Spontaneous Motility of Isolated Human Ureter

Slobodan M. Jankovic, Dobrivoje Stojadinovic, Miroslav Stojadinovic, Snezana V. Jankovic, Janko M. Djuric, Isidora Stojic, Marina Kostic

Short Communication

Biodistribution and Pharmacokinetic Study of 3,3′ Diseleno Dipropionic Acid (DSePA), A Synthetic Radioprotector, in Mice

Vikram Gota, Jayant S. Goda, Kartik Doshi, Anand Patil, Suvarna Sunderajan, Kiran Kumar, Mahendra Varne, Amit Kunwar, Vimal Kumar Jain, Indira Priyadarshini