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European Journal of Drug Metabolism and Pharmacokinetics

Issue 4/2016

Content (17 Articles)

Review Article

Regulations of Xenobiotics and Endobiotics on Carboxylesterases: A Comprehensive Review

Yanjiao Xu, Chengliang Zhang, Wenxi He, Dong Liu

Open Access Original Paper

Pharmacokinetics of mycophenolate sodium co-administered with tacrolimus in the first year after renal transplantation

Joanna Sobiak, Matylda Resztak, Maciej Głyda, Paulina Szczepaniak, Maria Chrzanowska

Original Paper

Pomegranate juice does not affect the disposition of simvastatin in healthy subjects

Soo-Jin Park, Chang-Woo Yeo, Eon-Jeong Shim, Hyunmi Kim, Kwang-Hyeon Liu, Jae-Gook Shin, Ji-Hong Shon

Original Paper

Population pharmacokinetic modeling of oxcarbazepine active metabolite in Chinese patients with epilepsy

Yunli Yu, Quanying Zhang, Wenjun Xu, Chengzhe Lv, Gang Hao

Original Paper

Pharmacokinetics, safety, and tolerability of rotigotine transdermal system in healthy Japanese and Caucasian subjects following multiple-dose administration

Willi Cawello, Seong Ryul Kim, Marina Braun, Jan-Peer Elshoff, Takeuchi Masahiro, Junji Ikeda, Tomoo Funaki

Original Paper

Population Pharmacokinetics and Pharmacodynamics of Piperacillin/Tazobactam in Patients with Nosocomial Infections

Rong Chen, Qing Qian, Meng-ru Sun, Chun-yan Qian, Su-lan Zou, Ming-li Wang, Li-ying Wang

Original Paper

Pharmacokinetics, Pharmacodynamics, and Tolerability of Single and Multiple Doses of Trandolapril, an Effective Angiotensin-Converting Enzyme Inhibitor, in Healthy Chinese Subjects

Xiaojiao Li, Chang Liu, Min Wu, Hong Zhang, Yanfu Sun, Longmei Cheng, Hong Chen, Chengjiao Liu, Lizhi Yang, Qi Zhang, Yuchen Cao, Jingkai Gu, Yanhua Ding

Original Paper

Genetic Determinants of Methotrexate Toxicity in Tunisian Patients with Rheumatoid Arthritis: A Study of Polymorphisms Involved in the MTX Metabolic Pathway

Souhir Chaabane, Sameh Marzouk, Rim Akrout, Mariem Ben Hamad, Yosser Achour, Ahmed Rebai, Leila Keskes, Hela Fourati, Zouhir Bahloul, Abdellatif Maalej

Original Paper

Prediction of the pharmacokinetics and tissue distribution of levofloxacin in humans based on an extrapolated PBPK model

Liqin Zhu, Yuan Zhang, Jianwei Yang, Yongming Wang, Jianlei Zhang, Yuanyuan Zhao, Weilin Dong

Open Access Original Paper

Physiologically based modeling of lisofylline pharmacokinetics following intravenous administration in mice

Elżbieta Wyska, Artur Świerczek, Krzysztof Pociecha, Katarzyna Przejczowska-Pomierny

Original Paper

Preparation, characterization and in vitro/vivo evaluation of tectorigenin solid dispersion with improved dissolution and bioavailability

Shuping Shuai, Shanlan Yue, Qingting Huang, Wei Wang, Junyi Yang, Ke Lan, Liming Ye

Original Paper

A pharmacokinetic study of patchouli alcohol after a single oral administration of patchouli alcohol or patchouli oil in rats

Ruoqi Zhang, Peiao Yan, Yunxia Li, Liang Xiong, Xiaohong Gong, Cheng Peng

Original Paper

Influence of Verapamil on Pharmacokinetics of Triptolide in Rats

Yichuan Zhang, Jin Li, Xiaolin Lei, Tianying Zhang, Guangxian Liu, Maohui Yang, Min Liu

Short Communication

Impact of a high-cholesterol diet on expression levels of Niemann–Pick C1-like 1 and intestinal transporters in rats and mice

Atsushi Kawase, Yasuha Araki, Yukiko Ueda, Sayaka Nakazaki, Masahiro Iwaki

Short Communication

Metabolic behavior prediction of pazopanib by cytochrome P450 (CYP) 3A4 by molecular docking

Xing-Jie Liu, Hua Lu, Ju-Xiang Sun, Su-Rong Wang, Yan-Shuai Mo, Xing-Sheng Yang, Ben-Kang Shi