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European Journal of Drug Metabolism and Pharmacokinetics

Issue 1/2017

Content (20 Articles)

Review Article

Enhancing Oral Absorption of β-Lapachone: Progress Till Date

Marival Bermejo, Victor Mangas-Sanjuan, Isabel Gonzalez-Alvarez, Marta Gonzalez-Alvarez

Original Research Article

External Validation of a Recently Developed Population Pharmacokinetic Model for Hydromorphone During Postoperative Pain Therapy

Harald Ihmsen, Doris Rohde, Jürgen Schüttler, Christian Jeleazcov

Original Research Article

Effect of Lactobacillus casei on the Pharmacokinetics of Amiodarone in Male Wistar Rats

Zuzana Matuskova, Pavel Anzenbacher, Rostislav Vecera, Michal Siller, Helena Tlaskalova-Hogenova, Jan Strojil, Eva Anzenbacherova

Original Research Article

Pharmacokinetic Studies of Oxathio-Heterocycle Fused Chalcones

Krystyna Okoniewska, Marek T. Konieczny, Krzysztof Lemke, Tomasz Grabowski

Open Access Original Research Article

Ocular Drug Distribution After Topical Administration: Population Pharmacokinetic Model in Rabbits

Nassim Djebli, Sonia Khier, Florence Griguer, Anne-Laure Coutant, Alexandra Tavernier, Gerard Fabre, Caroline Leriche, David Fabre

Original Research Article

Population Pharmacokinetics Modeling of Inhaled Umeclidinium for Adult Patients with Asthma

Shuying Yang, Laurie Lee, Steven Pascoe

Original Research Article

Inhibitory Effects of Triptolide on Human Liver Cytochrome P450 Enzymes and P-Glycoprotein

Hanhua Zhang, Guangkui Ya, Hongbing Rui

Open Access Original Research Article

Impact of CYP3A4*1G Allele on Clinical Pharmacokinetics and Pharmacodynamics of Clopidogrel

Dorota Danielak, Marta Karaźniewicz-Łada, Karolina Wiśniewska, Piotr Bergus, Paweł Burchardt, Anna Komosa, Franciszek Główka

Original Research Article

Pharmacokinetics, Safety and Tolerability of Sacubitril/Valsartan (LCZ696) After Single-Dose Administration in Healthy Chinese Subjects

Yi Han, Surya Ayalasomayajula, Wei Pan, Fan Yang, Yaozong Yuan, Thomas Langenickel, Markus Hinder, Sampath Kalluri, Parasar Pal, Gangadhar Sunkara

Original Research Article

Identification of Transporters Involved in Beraprost Sodium Transport In Vitro

Keiyu Oshida, Masahiro Shimamura, Kazuhiro Seya, Akihiro Ando, Yohei Miyamoto

Short Communication

Absolute Bioavailability of Ponesimod, a Selective S1P1 Receptor Modulator, in Healthy Male Subjects

Margaux Boehler, Pierre-Eric Juif, Matthias Hoch, Jasper Dingemanse

Short Communication

Pharmacokinetics of Saquinavir Mesylate from Oral Self-Emulsifying Lipid-Based Delivery Systems

Thiago Caon, Jadel Muller Kratz, Gislaine Kuminek, Melina Heller, Gustavo Amadeu Micke, Bibiana Verlindo de Araujo, Letícia Scherer Koester, Cláudia Maria Oliveira Simões

Short Communication

Pharmacokinetics of Oral and Intravenous Oseltamivir Treatment of Severe Influenza B Virus Infection Requiring Organ Replacement Therapy

Katharina Karsch, Xi Chen, Oliver Miera, Björn Peters, Patrick Obermeier, Roland C. Francis, Válerie Amann, Susanne Duwe, Pieter Fraaij, Alla Heider, Marcel de Zwart, Felix Berger, Albert Osterhaus, Brunhilde Schweiger, Barbara Rath