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Clinical Pharmacokinetics

Issue 5/2016

Content (9 Articles)

Open Access Review Article

Development of Human Membrane Transporters: Drug Disposition and Pharmacogenetics

Miriam G. Mooij, Anne T. Nies, Catherijne A. J. Knibbe, Elke Schaeffeler, Dick Tibboel, Matthias Schwab, Saskia N. de Wildt

Open Access Original Research Article

Effects of Age, Sex, and Race on the Safety and Pharmacokinetics of Single and Multiple Doses of Azilsartan Medoxomil in Healthy Subjects

Robert E. Harrell, Aziz Karim, Wencan Zhang, Caroline Dudkowski

Original Research Article

Use of Multiple Probes to Assess Transporter- and Cytochrome P450-Mediated Drug–Drug Interaction Potential of the Pangenotypic HCV NS5A Inhibitor Velpatasvir

Erik Mogalian, Polina German, Brian P. Kearney, Cheng Yong Yang, Diana Brainard, John McNally, Lisa Moorehead, Anita Mathias

Original Research Article

Pharmacokinetics of the Soluble Guanylate Cyclase Stimulator Riociguat in Healthy Young Chinese Male Non-Smokers and Smokers: Results of a Randomized, Double-Blind, Placebo-Controlled Study

Xia Zhao, Zining Wang, Yukun Wang, Hong Zhang, Hartmut Blode, Kenichi Yoshikawa, Corina Becker, Sigrun Unger, Reiner Frey, Yimin Cui

Original Research Article

Clinical Pharmacokinetics of Dulaglutide in Patients with Type 2 Diabetes: Analyses of Data from Clinical Trials

Jeanne S. Geiser, Michael A. Heathman, Xuewei Cui, Jennifer Martin, Corina Loghin, Jenny Y. Chien, Amparo de la Peña